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Ibicuruzwa

Methylophiopogonanone B.

Ibisobanuro bigufi:

Izina rusange: methylophiopogonone B.

Izina ry'icyongereza: methylophiopogonone B.

CAS No.: 74805-91-7

Uburemere bwa molekuline: 328.359

Ubucucike: 1.285

Ingingo yo guteka: 554.5 ± 49.0 ° C kuri 760 mmHg

Inzira ya molekulari: C19H20O5

Ingingo yo gushonga: N / A.

MSDS: N / A.

Ingingo ya Flash: 201.5 ± 23.3 ° C.


Ibicuruzwa birambuye

Ibicuruzwa

Gukoresha Methylophiopogonanone B.

Methylophiopogonone B, isodihydroflavone nyinshi, yakuwe mu mizi ya Ophiopogon japonicus, ifite antioxydants nyinshi.Methylophiopogonone B yongera GTP Rho kandi ikora binyuze muri Rho yerekana inzira.Methylophiopogonone B itera ihinduka ryimiterere yimikorere ya selile, harimo kugabanuka kwa dendritic no guhagarika fibre, binyuze muri actin cytoskeleton.

Izina rya Methylophiopogonanone B.

Izina ry'icyongereza:
(3R) -5,7-Dihydroxy-3 -

Igikorwa cyibinyabuzima cya Methylophiopogonanone B.

Ibisobanuro: methylophiopogonone B, isodihydroflavone ndende, yakuwe mu mizi ya Ophiopogon japonicus, ifite ubushobozi bwa antioxydeant.Methylophiopogonone B yongera GTP Rho kandi ikora binyuze muri Rho yerekana inzira.Methylophiopogonone B itera ihinduka ryimiterere yimikorere ya selile, harimo kugabanuka kwa dendritic no guhagarika fibre, binyuze muri actin cytoskeleton.

Ibyiciro bifitanye isano: umurima wubushakashatsi >> ibindi

inzira yerekana inzira >> G protein ihujwe na reseptor /

G protein >> RAS

Reba: [1] Wang Y, n'abandi.Homoisoflavonoids na Antioxidant

Igikorwa cya Ophiopogon japonicus Imizi.

Ito Y, n'abandi.Umukozi mushya, methylophiopogonanone B,

iteza imbere Rho gukora na tubulin depolymerisation.Ingirabuzimafatizo ya selile.2007 Werurwe;297 (1-2): 121-9.Epub 2006 Ukwakira 7.

Imiterere ya fiziki ya chimique ya Methylophiopogonanone B.

Ubucucike: 1.285

Ingingo yo guteka: 554.5 ± 49.0 ° C kuri 760 mmHg

Inzira ya molekulari: C19H20O5

Uburemere bwa molekuline: 328.359

Ingingo yerekana: 201.5 ± 23.3 ° C.

Misa nyayo: 328.131073

PSA : 75.99000

LogP : 5.22

Umuvuduko wamazi: 0.0 ± 1,6 mmHg kuri 25 ° C.

Igipimo cyangiritse: 1.617

Yongjian Service

Serivisi yihariye Yibikoresho Byifashishwa mubuvuzi gakondo bwabashinwa
Jiangsu Yongjian Pharmaceutical Technology Co., Ltd akora cyane cyane mubushakashatsi bwibanze bwibintu bikora byubuvuzi gakondo bwabashinwa mumyaka irenga icumi.Kugeza ubu, isosiyete imaze gukora ubushakashatsi bwimbitse ku bwoko burenga 100 bw’imiti gakondo ikoreshwa mu Bushinwa, kandi ikuramo ibihumbi n’ibigize imiti.

Isosiyete ifite abakozi bakuru ba R & D nibikoresho byiza byo gupima no gusesengura mu nganda, kandi imaze gukorera ibigo byubushakashatsi amagana.Irashobora kwihuta kandi neza ibyifuzo byabakiriya

Gutandukanya Ibiyobyabwenge, Gutegura no Kwemeza Serivisi
Umwanda mubi biyobyabwenge bifitanye isano rya bugufi nubwiza, umutekano n’umutekano w’ibiyobyabwenge.Gutegura no kwemeza imiterere yanduye mu biyobyabwenge birashobora kudufasha kumva inzira zanduye kandi bigatanga umusingi wo kunoza imikorere.Kubwibyo, gutegura no gutandukanya umwanda bifite akamaro kanini mubushakashatsi bwibiyobyabwenge niterambere.

Nyamara, ibirimo umwanda uri mu biyobyabwenge ni bike, isoko ni nini, kandi imiterere isa cyane ningenzi.Ni ubuhe buryo bw'ikoranabuhanga bwakoreshwa mu gutandukanya no kweza umwanda wose uri mu biyobyabwenge umwe umwe kandi vuba?Ni ubuhe buryo n'uburyo bukoreshwa mu kwemeza imiterere y'iyi myanda?Ngiyo ingorane ningorabahizi byugarije imiti myinshi yimiti, cyane cyane imishinga yimiti yubuvuzi bwibimera nubuvuzi bwa patenti mubushinwa.

Hashingiwe kubyo bikenewe, isosiyete yatangije serivisi zo gutandukanya no kwanduza ibiyobyabwenge.Isosiyete ishingiye kuri magnetiki resonance, mass spectrometrie nibindi bikoresho na tekinoroji, isosiyete irashobora kumenya byihuse imiterere yibintu bitandukanijwe, kugirango ibone ibyo abakiriya bakeneye.

Ubushakashatsi bw'inyamaswa
Ubuso bwubatswe bwahantu ho kugerageza inyamaswa ni metero kare 1500, harimo metero kare 400 zubushakashatsi bwa SPF kurwego na metero kare 100 za laboratoire ya P2.Iyobowe nabahanga bo muri kaminuza yimiti yubushinwa, ikora itsinda ryibanze rya tekinike hamwe nabatahutse.Tanga icyitegererezo cyiza cyinyamanswa, igishushanyo mbonera, imishinga rusange nizindi serivisi zubushakashatsi bwa siyanse yubumenyi bwibinyabuzima, kwigisha no guteza imbere inganda.

Umubare w'ubucuruzi

1. Kugaburira amatungo mato

2. Kwerekana indwara zinyamaswa

3. Gutanga umushinga wa kaminuza

4. Isuzuma rya farumasi muri vivo

5. Isuzuma rya farumasi

6. Serivisi yo kugerageza selile

Imbaraga zacu

1. Wibande ku bushakashatsi nyabwo

2. Kuringaniza byimazeyo inzira

3. Shyira umukono kumasezerano yibanga

4. Laboratoire yawe idafite aho ihurira

5. Itsinda rya tekinike yabigize umwuga ryemeza ubuziranenge bwubushakashatsi

SPF ibidukikije byubushakashatsi, byagenwe byabantu kugaburira, igihe-gikurikirana iterambere ryikigereranyo


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